Doxycycline analogues

Doxycycline inonzi semisynthetic antibiotic ine maitiro akawanda akaitwa, ari muboka re tetracyclines. Inogadzirwa nevakagadziri vakasiyana-siyana mumhando dzakasiyana-siyana dzekurapa:

Pharmacological action antibiotic Doxycycline

Mishonga inorwisa mabhakitiriya iri mubvunzo inoita nekudzivisa kupindirana kwemapuroteni mumasero ezvirwere zvehutachiona, sechikonzero chekuti ma microbes anorasikirwa nebasa ravo uye kukwanisa kubereka. Inopesana nemakorokoromu aya anotevera:

Minorganisms inoratidza kushorwa ne doxycycline:

Kupinda mumuviri, mishonga inorwisa mabhakitiriya inoparadzirwa mumasukisi uye mumhepo. Kurapa kwemishonga yemishonga inowanikwa muropa, mapapu, mapfupa, spleen, exudate ye sinasana paranasal, bile, maziso maziso pashure pehafu yeawa mushure mekutonga. Mumvura yomupfupa inopinda mumuto maduku. Iyo yakanyanyisa kubva mumuviri ine antibiotic ine nyota uye urini.

Zviratidzo zvekugadzwa kwaDoxycycline:

Chii chinogona kutora Doxycycline?

Muchirevo chekuti, mifananidzo yeDixycycline inenge mishonga yose yemishonga inonzi tetracycline-yakagadzirirwa inotevera :

Iyi mishonga inoratidzika nenzira yakadaro yeantimicrobial action uye inenge yakafanana nemishonga yemasikirwo. Kune zvishoma chete zvakasiyana zvinosanganiswa nezviratidzo zvekudya uye metabolism.

Doxycycline chinhu chinotorwa nemishonga inorwisa mabhakitiriya yematrocytine chaiyo, iyo inobudiswa nehuwandu hwemhando yefungus. Panguva imwe chete, nokuda kwehutano uye kuchengeteka kwemuviri, doxycycline inopfuura kupfuura "mutevedzeri" wayo. Kutenda kumakemikari, huwandu hwakawanda hwekunatswa kwemishonga inorwisa mabhakitiriya inogadziriswa, semugumisiro wekuti zviri nani kupinda uye zvinokwanisa kukonzera zvishoma nezvigumisiro. Doxycycline pasi pemamwe tetracycline mishonga inoderedza maruva anobatsira maruva, inozivikanwa nekugadzirisa zvakakwana uye nguva yakareba yekuita. Nokudaro, kushandiswa kwayo kunonyanya kuwedzerwa.

Mukuwedzera, Doxycycline inowanikwa mumhando dzakasiyana-siyana:

Pakati pedu zvakanyanya kupararira ndiyo fomu yekutanga inowanikwa pamisika yepamusoro pemapurisa nemagadziro akadaro, se:

Asi, zvinosuruvarisa, dioxycycline hydrochloride paanotorwa nemuromo kana paine kunonoka mune demo (semuenzaniso, nekuda kweatomical zvikamu) zvinogadzira acidification yakajeka yezvakatipoteredza. Izvi zvinokonzera kukuvadzwa kwemukati membrane, kusvika kune zvinoitika uye zvironda.

Nhoroondo yemazuva ano yemishonga inobva pa doxycycline - Unidox Solutab. Ichi chirwere chinosanganisira doxycycline monohydrate, iyo iyo yakasanganiswa haina kukonzera kuwedzera mu acidity uye inowanikwa mumatomu emagumisi inenge yakakwana zvachose. Panguva imwecheteyo, mucous membrane haitambudzi, hapana chinhu chinokonzera pamatumbo microflora, uye mikana yekuvandudza dyspeptic phenomena haigoni. Iyo inyanzvi inogona kuparara mumvura, kuwana kumira, iyo isingabatanidzi kukanganisa kwayo kunonoka.